PG 106 acetate
Cat# NB-64-68588-25mg
Size : 25mg
Brand : Neo Biotech
PG 106 acetate (Synonyms: PG 106 acetate(944111-22-2 Free base))
Catalog No. TP1952L Copy Product Info
Purity: 99.93%
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM.
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Purity:99.93%
Appearance:Solid
Color:White
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM. |
| Targets&IC50 | MC3R (human):210 nM |
| Synonyms | PG 106 acetate(944111-22-2 Free base) |
| Molecular Weight | 1068.23 |
| Formula | C53H73N13O11 |
| Smiles | CCCCC(NC(C)=O)C(N[C@H]1CC(NCCCC[C@@H](C(N)=O)NC([C@H](CC2=CNC3=CC=CC=C32)NC([C@H](CCC/N=C(N)\N)NC([C@@H](CC4=CC5=CC=CC=C5C=C4)NC(CCNC1=O)=O)=O)=O)=O)=O)=O.CC(O)=O |
| Sequence | Ac-DL-Nle-Asp(1)-bAla-D-2Nal-Arg-Trp-Lys(1)-NH2 |
| Sequence Short | {Nle}-D-{Bal}-{D-Nal}-RWK (Lactam bridge:Asp2-Lys7) |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature. |


