PG 106 acetate

Referência NB-64-68588-25mg

Tamanho : 25mg

Marca : Neo Biotech

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PG 106 acetate (Synonyms: PG 106 acetate(944111-22-2 Free base))

Catalog No. TP1952L Copy Product Info
Purity: 99.93%
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM.

PG 106 acetate

Copy Product Info
Synonyms PG 106 acetate(944111-22-2 Free base)

PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM.

PG 106 acetate
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Purity:99.93%
Appearance:Solid
Color:White
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Product Introduction

Bioactivity
Description
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM.
Targets&IC50
MC3R (human):210 nM
SynonymsPG 106 acetate(944111-22-2 Free base)
Chemical Properties
Molecular Weight1068.23
FormulaC53H73N13O11
SmilesCCCCC(NC(C)=O)C(N[C@H]1CC(NCCCC[C@@H](C(N)=O)NC([C@H](CC2=CNC3=CC=CC=C32)NC([C@H](CCC/N=C(N)\N)NC([C@@H](CC4=CC5=CC=CC=C5C=C4)NC(CCNC1=O)=O)=O)=O)=O)=O)=O.CC(O)=O
SequenceAc-DL-Nle-Asp(1)-bAla-D-2Nal-Arg-Trp-Lys(1)-NH2
Sequence Short{Nle}-D-{Bal}-{D-Nal}-RWK (Lactam bridge:Asp2-Lys7)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature.